Cyproterone acetate (CPA), sold alone under the brand name Androcur or with ethinylestradiol under the brand names Diane or Diane-35 among others, is an antiandrogen and progestin medication used in the treatment of androgen-dependent conditions such as acne, excessive body hair … See more CPA is used as a progestin and antiandrogen in hormonal birth control and in the treatment of androgen-dependent conditions. Specifically, CPA is used in combined birth control pills, in the treatment of … See more CPA is generally well-tolerated and has a mild side-effect profile regardless of dosage when it is used in combination with an estrogen in women. Side effects of CPA in general include hypogonadism (low sex-hormone levels) and associated symptoms such as See more Inhibitors and inducers of the cytochrome P450 enzyme CYP3A4 may interact with CPA. Examples of strong CYP3A4 inhibitors include See more CPA, also known as 1α,2α-methylene-6-chloro-17α-acetoxy-δ -progesterone or as 1α,2α-methylene-6-chloro-17α-hydroxypregna-4,6-diene-3,20-dione acetate, is a synthetic pregnane steroid and an acetylated derivative of 17α-hydroxyprogesterone. … See more Contraindications of CPA include: • Hypersensitivity to CPA or any of the other components of the medication • Pregnancy, lactation, and breastfeeding • Puberty (except if being used to treat precocious puberty or delay puberty) See more CPA is relatively safe in acute overdose. It is used at very high doses of up to 300 mg/day by mouth and 700 mg per week by intramuscular … See more Pharmacodynamics CPA has antiandrogenic activity, progestogenic activity, weak partial glucocorticoid activity, weak steroidogenesis inhibitor activity, and agonist activity at the pregnane X receptor. It has no See more WebJun 15, 2024 · Cyproterone - an anti-androgen for men Cyprostat, Androcur. Cyproterone - an anti-androgen for men. Take cyproterone tablets with a drink of water and something to eat. Cyproterone may make you feel tired or weak. If this happens, do not drive and do not use tools or machines. Cyproterone can affect the way your liver works and the way …
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WebCyproterone acetate C24H29ClO4 - PubChem Apologies, we are having some trouble retrieving data from our servers... PUGVIEW FETCH ERROR: 403 Forbidden National … WebFeb 14, 2024 · The possibility of suboptimal breast development with progestogens is of particular relevance to cyproterone acetate (CPA; Androcur). This is because cyproterone acetate is a potent progestogen in addition to antiandrogen and is used in transfeminine people at doses that result in very strong progestogenic exposure . flyers anime
Side effects of cyproterone acetate - Wikipedia
WebThe combination of ethinyl estradiol and cyproterone acetate results in maximal suppression of serum testosterone levels and blocking of the androgen receptor. 1 TABLE 1: Results of case reports of the histologic changes induced in the mammary gland of male-to-female transsexuals WebWhat will it do for me? This medication contains a combination of two ingredients: cyproterone and ethinyl estradiol. Cyproterone belongs to a group of medications known as antiandrogens. Ethinyl estradiol belongs to a group of medications known as estrogens. WebHydrocortisone is the pharmaceutical term for cortisol used in oral administration, intravenous injection, or topical application. It is used as an immunosuppressive drug, given by injection in the treatment of severe … green irrigation long island